Skip to main content
U.S. flag

An official website of the United States government

Here’s how you know

Dot gov

Official websites use .gov
A .gov website belongs to an official government organization in the United States.

HTTPS

Secure .gov websites use HTTPS
A lock ( Lock A locked padlock ) or https:// means you’ve safely connected to the .gov website. Share sensitive information only on official, secure websites.

  • Environmental Topics
  • Laws & Regulations
  • Report a Violation
  • About EPA
Risk Assessment
Contact Us

Breaking the Barrier: Using Novel In Vitro Organotypic Airway Trans-Epithelial Exposure Model to Study the Depth and Dynamics of Inhaled Chemical Toxicity

On this page:

  • Overview
Inhaled chemical testing and research have focused heavily on airway epithelial cells; however, there are a diverse range of other lung cell types within the cellular microenvironment whose role as targets and/or mediators of exposure effects are poorly understood. While one such cell type, the lung fibroblast, occupies a large percentage of the respiratory tract tissue volume and plays a critical role in regulating tissue homeostasis, we know very little about its role as a target and/or mediator of adverse exposure effects. To address this knowledge gap, we developed in vitro organotypic models that recapitulate in vivo exposure of the airway microenvironment by incorporating a functional human bronchial epithelial cell (HBEC) barrier to separate human lung fibroblasts (HLF) from the inhaled exposure material. The model design allows also for the assessment of direct and trans-epithelial effects of toxicant exposure in the HBEC and HLF, respectively, in parallel to provide insight into the roles that these different cell types within the airway microenvironment play in the effects of inhaled chemical exposures. Using this model, we identified the molecular dynamics of direct and trans-epithelial oxidative stress and induction of a pro-inflammatory state including intracellular ROS accumulation, glutathione oxidation, cellular signaling pathway activation, NRF2 signaling, and gene expression at the RNA and protein levels. Trans-epithelial DEP and WS exposures caused oxidative stress as well as oxidative stress-responsive and pro-inflammatory gene expression in HLF. The effects of trans-epithelial DEP and WS exposure on fibroblasts were similar to, or greater than, those observed in adjacent directly exposed HBEC. We also determined that pre-treatment of HLF with antioxidants augments the oxidative stress response in both HLF and HBEC. Our findings indicate that inhaled oxidants have trans-epithelial effects on HLF, suggest that HLF are more susceptible to oxidative injury than HBEC, and demonstrate that HLF mediate the effects of direct inhaled oxidant exposure in adjacent HBEC. These observations illustrate the prospective benefit of improving the physiological relevance of in vitro models and examining the potential for trans-epithelial exposure effects in inhaled chemical research and testing. Does not reflect EPA policy.

Impact/Purpose

To present research describing the development and use of novel in vitro NAMs for assessing the trans-epithelial and trans-alveolar effects of inhaled chemical exposures in chemical research and testing.

Citation

McCullough, S. Breaking the Barrier: Using Novel In Vitro Organotypic Airway Trans-Epithelial Exposure Model to Study the Depth and Dynamics of Inhaled Chemical Toxicity. Virtual-South Central Society of Toxicology Regional Chapter Meeting, Virtual, Virtual, November 13, 2020.
  • Risk Assessment Home
  • About Risk Assessment
  • Risk Recent Additions
  • Human Health Risk Assessment
  • Ecological Risk Assessment
  • Risk Advanced Search
    • Risk Publications
  • Risk Assessment Guidance
  • Risk Tools and Databases
  • Superfund Risk Assessment
  • Where you live
Contact Us to ask a question, provide feedback, or report a problem.
Last updated on March 03, 2021
United States Environmental Protection Agency

Discover.

  • Accessibility Statement
  • Budget & Performance
  • Contracting
  • EPA www Web Snapshots
  • Grants
  • No FEAR Act Data
  • Privacy
  • Privacy and Security Notice

Connect.

  • Data
  • Inspector General
  • Jobs
  • Newsroom
  • Open Government
  • Regulations.gov
  • Subscribe
  • USA.gov
  • White House

Ask.

  • Contact EPA
  • EPA Disclaimers
  • Hotlines
  • FOIA Requests
  • Frequent Questions

Follow.